WebNov 12, 2024 · Multicomponent reactions (MCRs) are very important to provide enantiomerically enriched compounds with high structural diversity and complexity. These reactions play an important role in the synthesis of natural products, commercial drugs, agrochemicals and catalysts. Currently, CPA-catalyzed enantioselective MCRs are a hot … WebApr 12, 2024 · We have developed a chiral phosphoric acid-catalyzed enantioselective Friedel–Crafts alkylation reaction between pyrroles and indolylmethanols. Wide …
Mukaiyama Michael Reaction - an overview ScienceDirect Topics
WebMay 4, 2007 · Mannich-type reaction of ketene silyl acetals with aldimines proceeded catalytically by means of a phosphoric acid diester, derived from (R)-BINOL, as a chiral Brønsted acid to afford β-amino esters with good diastereoselectivity in favor of the syn isomer and high enantioselectivity (up to 96% ee).The highest enantioselectivity was … WebJun 5, 2024 · An enantioselective intramolecular anti-SN2′ cyclization reaction for the construction of a quaternary stereogenic center was accomplished through the activation of the leaving group using a binaphthol-derived phosphoramide as the chiral Brønsted acid catalyst. The present allylic substitution reaction is be 2024 Chemical Science HOT … simon williamson clinic birmingham
Enantioselective transition metal catalysis directed by chiral …
WebApr 8, 2024 · The first copper-catalyzed atroposelective Michael-type addition between azonaphthalenes and arylboronic acids for the construction of biaryl atropisomers was established using a novel BINOL-derived phosphoramidite as a chiral ligand. A broad range of atropisomeric biaryls were obtained with good efficiency, and the practicality of this … WebReactions that form a new chiral center If the starting material is achiral, then we will always get a racemic mixture of our product enantiomers, unless some other chiral agent is involved. This is for the same reason … WebA new strategy of asymmetric carbonyl catalysis via a chiral Lewis acid-bonded aldehyde has been developed for the direct Mannich/condensation cascade reaction of glycine ester with aromatic aldimines. The co-catalytic system of 2-picolinaldehyde and chiral Yb III-N,N′-dioxides was identified to be efficient under mild conditions, providing a series of … simon williams ttuhsc